Product Size
25 mg
5 mg
Custom Size
Product Overview
Description
Potent, competitive, selective and cell-permeable inhibitor of CaM-KK.
Biological Description
Potent, competitive, selective and cell-permeable inhibitor of CaM-KK (Ki values are0.21 µM and 40 nM for CaM-KKα and CaM-KKβ respectively). Potent, competitive AhR agonist (EC50 = 43 nM). Active in vivo.
Solubility Overview
Soluble in DMSO to 25 mM.
Chemical Properties
Chemical Name
7-Oxo-7H-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acid acetate
Molecular Weight (Da)
374.35
Molecular Formula
C19H10N2O3.C2H4O2
SMILES
CC(=O)O.C1=CC=C2C(=C1)N=C3N2C(=O)C4=CC=CC5=C(C=CC3=C54)C(=O)O
Storage & Handling
Storage Instructions
Store at room temperature. The product can be stored for up to 12 months.
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20 °C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
