Product Size
5 mg
25 mg
Custom Size
Product Overview
Description
An inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3.
Biological Description
PFK158 is an inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3; IC50 = 137 nM for human recombinant PFKFB3).
Solubility Overview
Soluble in DMSO to 75 mM.
Chemical Properties
Chemical Name
(E)-1-pyridin-4-yl-3-[7-(trifluoromethyl)quinolin-2-yl]prop-2-en-1-one
Molecular Weight (Da)
328.30
Molecular Formula
C18H11F3N2O
SMILES
C1=CC(=CC2=C1C=CC(=N2)C=CC(=O)C3=CC=NC=C3)C(F)(F)F
Storage & Handling
Storage Instructions
Shipped at 4 °C. Store at -20 °C.
